Docking 14 Million Virtual Isoquinuclidines against the µ and ? Opioid Receptors Reveals Dual Antagonists–Inverse Agonists with Reduced Withdrawal Effects.

Seth F. Vigneron, Shohei Ohno, Joao Braz, Joseph Y. Kim, Oh Sang Kweon, Chase Webb, Christian B. Billesbølle, Karthik Srinivasan, Karnika Bhardwaj, John J. Irwin, Aashish Manglik, Allan I. Basbaum, Jonathan A. Ellman, Brian K. Shoichet. Docking 14 Million Virtual Isoquinuclidines against the µ and ? Opioid Receptors Reveals Dual Antagonists–Inverse Agonists with Reduced Withdrawal Effects. ACS Central Science. 2025 Apr 29.

2025
https://researcherprofiles.org/profile/613784770

Seth F. Vigneron, Shohei Ohno, Joao Braz, Joseph Y. Kim, Oh Sang Kweon, Chase Webb, Christian B. Billesbølle, Karthik Srinivasan, Karnika Bhardwaj, John J. Irwin, Aashish Manglik, Allan I. Basbaum, Jonathan A. Ellman, Brian K. Shoichet